1: With Dess-Martin periodane; sulfuric acid in dichloromethane T=0 - 25°C; 2: With sodium hydrogencarbonate in dichloromethane; water 0.333333 h; Product distribution / selectivity;
1: With 4-(N,N-dimethlyamino)pyridine in toluene T=20 - 70°C; 3 h; 2: With tert-butyl methyl ether in toluene T=10°C; 1 h; Product distribution / selectivity;
1: 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one With sodium hydride in N,N-dimethyl-formamide T=0°C; 2: n-hexadecanoyl chloride in N,N-dimethyl-formamide T=0°C; 5 h; Product distribution / selectivity;
