反应条件
1: p-bromophenyl mercaptan With sodium hydride in N,N-dimethyl-formamide 0.5 h; 2: benzyl bromide; 2-bromo-1-ethanol in N,N-dimethyl-formamide 20 h; Further stages.;
参考文献
Hajduk, Philip J.; Shuker, Suzanne B.; Nettesheim, David G.; Craig, Richard; Augeri, David J.; Betebenner, David; Albert, Daniel H.; Guo, Yan; Meadows, Robert P.; Xu, Lianhong; Michaelides, Michael; Davidsen, Steven K.; Fesik, Stephen W.
Journal of Medicinal Chemistry, 2002 , vol. 45, # 26 p. 5628 - 5639