反应条件
1.1: n-butyllithium / tetrahydrofuran / 1 h / -5 °C 1.2: 18 h / 50 °C 2.1: 3-chloro-benzenecarboperoxoic acid / ethylene glycol dimethyl ether / 7 h / 0 - 20 °C 3.1: methanesulfonyl chloride / N,N-dimethyl-formamide / 2 h / 60 °C View Scheme
参考文献
Liddle, John; Bamborough, Paul; Barker, Michael D.; Campos, Sebastien; Chung, Chun-Wa; Cousins, Rick P.C.; Faulder, Paul; Heathcote, Michelle L.; Hobbs, Heather; Holmes, Duncan S.; Ioannou, Chris; Ramirez-Molina, Cesar; Morse, Mary A.; Osborn, Ruth; Payne, Jeremy J.; Pritchard, John M.; Rumsey, William L.; Tape, Daniel T.; Vicentini, Giorgia; Whitworth, Caroline; Williamson, Rick A.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 16 p. 5222 - 5226