反应条件
1: 1) CuI, aq. NH4OH, NH2OH*HCl / 1) EtOH, 15 min, 2) DMF, 110 to 120 deg C, 3 h
2: 62 percent / 3percent aq. NaOH / ethanol / 2 h
View Scheme
参考文献
Defranq, Eric; Zesiger, Thierry; Tabacchi, Raffaele
Helvetica Chimica Acta, 1993 , vol. 76, # 1 p. 425 - 430