反应条件
1: 95 percent / NaN3, TFA / CHCl3 / a) 0 deg C, 1 h, b) r.t., 4 h 2: 85 percent / H2 / 10 percent Pd/C / ethanol / 24 h / 2585.7 Torr / Ambient temperature View Scheme
参考文献
Wey, Shiow-Jyi; O'Connor, Kenneth J.; Burrows, Cynthia J.
Tetrahedron Letters, 1993 , vol. 34, # 12 p. 1905 - 1908