反应条件
1: N-ethyl-N,N-diisopropylamine / 1,4-dioxane / 13 h / 100 °C
2: trifluoroacetic acid / dichloromethane / 20 °C
View Scheme
参考文献
Zhang, Zaihui; Sun, Shaoyi; Kodumuru, Vishnumurthy; Hou, Duanjie; Liu, Shifeng; Chakka, Nagasree; Sviridov, Serguei; Chowdhury, Sultan; McLaren, David G.; Ratkay, Leslie G.; Khakh, Kuldip; Cheng, Xing; Gschwend, Heinz W.; Kamboj, Rajender; Fu, Jianmin; Winther, Michael D.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 2 p. 568 - 583