N-(2-氰基-3-氟苯基)吡咯合成路线 (共 2 条)
反应条件
caesium carbonate in N,N-dimethyl-formamide T=80°C;
参考文献
JANSSEN PHARMACEUTICA NV; MEERPOEL, Lieven; MAES, Louis, Jules, Roger, Marie; DE WIT, Kelly
Patent: WO2012/84804 A1, 2012 ;
Location in patent: Page/Page column 54 ;
反应条件
acetic acid Hantzsch pyrrole synthesis; 0.5 h; Heating;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 15, # 14 p. 3453 - 3458