2-甲硫基-4,5-嘧啶二甲酸二乙酯合成路线 (共 4 条)
反应条件
sodium acetate; (1,1'-bis(diphenylphosphine)ferrocene)palladium(0) T=140°C; P=18751.9 Torr; Parr reactor;
参考文献
TIBOTEC PHARMACEUTICALS LTD.
Patent: WO2004/96807 A2, 2004 ;
Location in patent: Page 70 ;
反应条件
sodium acetate in N,N-dimethyl-formamide T=80 - 90°C; 12 h;
参考文献
Sansebastiano; Mosti; Menozzi; Schenone; Muratore; Petta; Debbia; Pesce Schito; Schito
Farmaco, 1993 , vol. 48, # 3 p. 335 - 355
反应条件
1: 0.5 h / 0 °C 2: sodium / ethanol / 1 h / Heating View Scheme
参考文献
Medicinal Chemistry Research, , vol. 10, # 1 p. 19 - 29
反应条件
sodium in ethanol 1 h; Heating;
参考文献
Medicinal Chemistry Research, , vol. 10, # 1 p. 19 - 29