反应条件
1: POCl3; ZnCl2 / 1,2-dichloro-ethane / 4 h / 70 °C 2: 1,1'-carbonyldiimidazole; K2CO3; DMAP / dimethylformamide / 4 h / 85 °C View Scheme
参考文献
McKie, Jeffrey A.; Bhagwat, Shripad S.; Brady, Helen; Doubleday, Mary; Gayo, Leah; Hickman, Mathew; Jalluri, Ravi K.; Khammungkhune, Sak; Kois, Adam; Mortensen, Deborah; Richard, Normand; Sapienza, John; Shevlin, Graziella; Stein, Bernd; Sutherland, May
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 13 p. 3407 - 3410