1: 3-methoxy-phenol With sodium hydride in tetrahydrofuran; mineral oil
T=20°C; 1 h; Cooling with ice;
2: bromomethyl-methyl-ether in tetrahydrofuran; mineral oil
T=20°C; 2 h;
参考文献
AUTIFONY THERAPEUTICS LIMITED; ALVARO, Giuseppe; DAMBRUOSO, Paolo; MARASCO, Agostino; TOMMASI, Simona; DECOR, Anne; LARGE, Charles
Patent: WO2012/76877 A1, 2012 ;
Location in patent: Page/Page column 81-82 ;
WO 2012/076877 A1