5-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯合成路线

5-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯合成路线（共 6 条）

2312-23-43-氯苯肼盐酸盐

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

参考文献

US4775409 A1, ;

2312-23-43-氯苯肼盐酸盐+

94-05-32-氰基-3-乙氧基丙烯酸乙酯

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

参考文献

Eli Lilly and Company
Patent: US4620865 A1, 1986 ;

42466-67-1(E)-2-氰基-3-乙氧基丙烯酸乙酯+

2312-23-43-氯苯肼盐酸盐

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

参考文献

BRISTOL-MYERS SQUIBB COMPANY; PINTO, Donald J.; CORTE, James R.; GILLIGAN, Paul J.; FANG, Tianan; SMITH II, Leon M.; WANG, Yufeng; YANG, Wu; EWING, William R.
Patent: WO2013/22818 A1, 2013 ;
Location in patent: Paragraph 00321 ;
WO 2013/022818 A1

14763-20-3间氯苯肼+

94-05-32-氰基-3-乙氧基丙烯酸乙酯

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

参考文献

Organic Letters, , vol. 15, # 19 p. 5044 - 5047

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

110821-39-15-溴-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

参考文献

Beck, James R.; Gajewski, Robert P.; Lynch, Michael P.; Wright, Fred L.
Journal of Heterocyclic Chemistry, 1987 , vol. 24, p. 267 - 270

15001-08-85-氨基-1-(3-氯苯基)-1H-吡唑-4-羧酸乙酯

98534-74-85-氯-1-（3-氯苯基）-1H-吡唑-4-羧酸乙酯

参考文献

Beck, James R.; Gajewski, Robert P.; Lynch, Michael P.; Wright, Fred L.
Journal of Heterocyclic Chemistry, 1987 , vol. 24, p. 267 - 270