反应条件
1: K2CO3 / ethanol; H2O / 24 h / 105 °C 2: dimethylformamide 3: 1.) H2, p-toluenesulfonic acid monohydrate, 2.) p-toluenesulfonic acid monohydrate / 1.) 10percent Pd/C / 1.) MeOH, 37 psi, 2 h, 2.) MeOH, 60 deg C, 1 h View Scheme
参考文献
TenBrink, Ruth E.; Im, Wha B.; Sethy, Vimala H.; Tang, Andrew H.; Carter, Don B.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 6 p. 758 - 768
