1: Et3N, methanesulfonyl chloride / CH2Cl2 / 24 h / Ambient temperature
2: tetra-n-butylammonium fluoride / tetrahydrofuran; diethyl ether / 0.17 h / Ambient temperature
View Scheme
参考文献
Woo, L. W. Lawrence; Howarth, Nicola M.; Purohit, Atul; Hejaz, Hatem A. M.; Reed, Michael J.; Potter, Barry V. L.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 7 p. 1068 - 1083