反应条件
1: 88 percent / 2N aq. KOH / 24 h / Ambient temperature
2: 1.) POCl3, 2.) 1N aq. HCl / 1.) reflux, 1 h, 2.) reflux, 1 h
3: 76 percent / K2CO3 / acetone
View Scheme
参考文献
Mongrain, Colette; Brassard, Paul
Heterocycles, 1993 , vol. 36, # 9 p. 2109 - 2128