1: para-bromoacetophenone With sodium hexamethyldisilazane in tetrahydrofuran T=0°C; 0.75 h; 2: 1-(trifluoroacetyl)-imidazole in tetrahydrofuran T=-78 - 20°C;
参考文献
Prabhakaran, Jaya; Majo, Vattoly J.; Simpson, Norman R.; Van Heertum, Ronald L.; Mann, J. John; Kumar, J. S. Dileep
Journal of Labelled Compounds and Radiopharmaceuticals, 2005 , vol. 48, # 12 p. 887 - 895