2-(四唑-5-基)苯硼酸合成路线 (共 2 条)
反应条件
1: With potassium hydroxide; palladium diacetate; triphenylphosphine in water; isopropyl alcohol; toluene T=70°C; 5 h; 2: in water; isopropyl alcohol; toluene T=20°C; pH=2; Acidic conditions;
参考文献
EP1777224 A2, ;
Page/Page column 7 ;
反应条件
potassium carbonate; palladium diacetate; triphenylphosphine in water; toluene T=60 - 70°C; 16 h; Product distribution / selectivity;
参考文献
QUIMICA SINTETICA, S.A.
Patent: WO2006/134078 A1, 2006 ;
Location in patent: Page/Page column 16 ;