反应条件
1: 4-amino-phenol With sodium hydride in N,N-dimethyl-formamide T=20°C; 0.5 h; 2: ethyl iodide in N,N-dimethyl-formamide T=20°C; 20 h; Further stages.;
参考文献
Xie, Hui; Ng, Danny; Savinov, Sergey N.; Dey, Barna; Kwong, Peter D.; Wyatt, Richard; Smith III, Amos B.; Hendrickson, Wayne A.
Journal of Medicinal Chemistry, 2007 , vol. 50, # 20 p. 4898 - 4908