反应条件
1: 32 percent / Et3N, KI / dimethylformamide / 72 h / Ambient temperature 2: 24 percent / H2, 3 N HCl / 10percent Pd/C / ethanol / 12 h / 50 °C / 3800 Torr 3: 70 percent / Et3N, KI / dimethylformamide / 72 h / Ambient temperature 4: 67 percent / H2, 3 N HCl / 10percent Pd/C / ethanol / 12 h / 50 °C / 3800 Torr View Scheme
参考文献
Melchiorre, Carlo; Bolognesi, Maria L.; Chiarini, Alberto; Minarini, Anna; Spampinato, Santi
Journal of Medicinal Chemistry, 1993 , vol. 36, # 23 p. 3734 - 3737
