1-(5-甲基吡啶-2-基)哌啶-4-醇合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in 1-methyl-pyrrolidin-2-one T=200°C; 1 h; microwave reactor;
参考文献
Mitsubishi Tanabe Pharma Corporation
Patent: EP2390254 A1, 2011 ;
Location in patent: Page/Page column 61 ;
EP 2390254 A1