反应条件
1: bis-triphenylphosphine-palladium(II) chloride; sodium carbonate / N,N-dimethyl-formamide; water / 0.1 h / 110 °C / |Microwave irradiation
2: carbon tetrabromide; triphenylphosphine / dichloromethane / 1.25 h / 0 - 20 °C
View Scheme
参考文献
PIRAMAL ENTERPRISES LIMITED; KUMAR, Sanjay; SHARMA, Rajiv; MAHAJAN, Vishal, Ashok; SAWARGAVE, Sangameshwar, Prabhakar
Patent: WO2013/128378 A1, 2013 ;