反应条件
1: palladium (II) acetate, triphenylarsine, triethylamine / various solvent(s) / 80 °C 2: 30percent NH3 MeOH, dioxane / Ambient temperature View Scheme
参考文献
Verlinde, Christophe L. M. J.; Callens, Mia; Calenbergh, Serge Van; Aerschot, Arthur Van; Herdewijn, Piet; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 21 p. 3605 - 3613