反应条件
1: (S)-1-{3-[(E)-2-(7-chloro-quinolin-2-yl)-vinyl]-phenyl}-3-[2-(1-hydroxy-1-methylethyl)-phenyl]-propan-1-ol With methanesulfonyl chloride; N-ethyl-N,N-diisopropylamine in tetrahydrofuran; toluene T=-15°C; 1 h; 2: methyl 2-(2-(sulfanylmethyl)cyclopropyl)acetate With caesium carbonate in tetrahydrofuran; N,N-dimethyl-formamide; toluene T=20°C;