反应条件
1: 1.) K2CO3, 2.) tetra-n-butylammonium iodide / 1.) DMF, 2.) DMF, RT 2: 11.5 mg / H2 / 10percent Pd-C / tetrahydrofuran / 2792.6 Torr View Scheme
参考文献
Cushman; He; Katzenellenbogen; Lin; Hamel
Journal of Medicinal Chemistry, 1995 , vol. 38, # 12 p. 2041 - 2049