1: With diphenyl phosphoryl azide; triethylamine in tert-butyl alcohol 6 h; Heating; 2: With hydrogenchloride in tetrahydrofuran 6 h; Heating;
参考文献
Padmanabhan, Seetharamaiyer; Perlman, Michael E; Zhang, Lu; Moore, Deke; Zhou, Dan; Fischer, James B; Durant, Graham J; McBurney, Robert N
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 4 p. 501 - 504