N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺合成路线 (共 2 条)
反应条件
in N,N-dimethyl-formamide 2 h;
参考文献
SEATTLE GENETICS, INC.
Patent: WO2007/8848 A2, 2007 ;
Location in patent: Page/Page column 108; 136; 137 ;
反应条件
N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide 1 h;
参考文献
WO2007/8603 A1, ;
Page/Page column 137; 166; 167 ;