反应条件
benzotriazol-1-ol; O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; N-ethyl-N,N-diisopropylamine in diethylene glycol dimethyl ether
T=100°C; 0.5 h; microwave irradiation;
参考文献
Santagada, Vincenzo; Frecentese, Francesco; Perissutti, Elisa; Cirillo, Donatella; Terracciano, Sara; Caliendo, Giuseppe
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 17 p. 4491 - 4493