(1S,2s)-(+)-反式-1-氨基-2-茚醇合成路线 （共 13 条）
反应条件
1: 91 percent / Et3N / dimethylformamide / 1 h / Ambient temperature 2: 92 percent / SOCl2 / CH2Cl2 / 3 h / Ambient temperature 3: 92 percent / 20percent H2SO4 / CH2Cl2 / 10 h / Heating View Scheme
参考文献
Lehr; Billich; Charpiot; Ettmayer; Scholz; Rosenwirth; Gstach
Journal of Medicinal Chemistry, 1996 , vol. 39, # 10 p. 2060 - 2067
反应条件
1: 91 percent / Et3N / dimethylformamide / 1 h / Ambient temperature 2: 92 percent / SOCl2 / CH2Cl2 / 3 h / Ambient temperature 3: 92 percent / 20percent H2SO4 / CH2Cl2 / 10 h / Heating View Scheme
参考文献
Lehr; Billich; Charpiot; Ettmayer; Scholz; Rosenwirth; Gstach
Journal of Medicinal Chemistry, 1996 , vol. 39, # 10 p. 2060 - 2067
反应条件
sodium carbonate in tetrahydrofuran; water
T=0 - 20°C; 3 h;
参考文献
Ren, Qiao; Siau, Woon-Yew; Du, Zhiyun; Zhang, Kun; Wang, Jian
Chemistry - A European Journal, 2011 , vol. 17, # 28 p. 7781 - 7785
