1-trifluoromethylsulfonyl-1H-1,2,3-benzotriazole multistep reaction; var. Grignard reagents and amines; var. reag. in 2.) step: Tf2O or Ac2O; Product distributionMechanism;
参考文献
Katritzky; Moutou; Yang
Synthesis, 1995 , # 12 p. 1497 - 1505
1: acetophenone With potassium tert-butylate in tetrahydrofuran
T=20°C; 0.5 h;
2: Pentanethioic acid benzylamide in tetrahydrofuran
T=20°C; 4 h; Further stages.;
参考文献
Katritzky, Alan R.; Khashab, Niveen M.; Haase, Danniebelle N.; Yoshioka, Megumi; Ghiviriga, Ion; Steel, Peter J.
Journal of Organic Chemistry, 2007 , vol. 72, # 18 p. 6742 - 6748
