Bach, Peter; Bostroem, Jonas; Brickmann, Kay; Van Giezen; Groneberg, Robert D.; Harvey, Darren M.; O'Sullivan, Michael; Zetterberg, Fredrik
European Journal of Medicinal Chemistry, 2013 , vol. 65, p. 360 - 375
1: 82 percent / 2 h / 135 °C
2: 97.7 percent / thionyl chloride / various solvent(s) / 1.5 h / 25 °C
3: 73 percent / NaI, K2CO3 / acetonitrile / 24 h / Heating
View Scheme
参考文献
Diana, Guy D.; Oglesby, Richard C.; Akullian, Vahan; Carabateas, Phillip M.; Cutcliffe, David; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 2 p. 383 - 388
1: 82 percent / 2 h / 135 °C
2: 97.7 percent / thionyl chloride / various solvent(s) / 1.5 h / 25 °C
3: 53 percent / NaI, K2CO3 / acetonitrile / 24 h / Heating
View Scheme
参考文献
Diana, Guy D.; Oglesby, Richard C.; Akullian, Vahan; Carabateas, Phillip M.; Cutcliffe, David; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 2 p. 383 - 388
1: 82 percent / 2 h / 135 °C
2: 97.7 percent / thionyl chloride / various solvent(s) / 1.5 h / 25 °C
3: 69 percent / NaI, K2CO3 / acetonitrile / 24 h / Heating
View Scheme
参考文献
Diana, Guy D.; Oglesby, Richard C.; Akullian, Vahan; Carabateas, Phillip M.; Cutcliffe, David; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 2 p. 383 - 388
