1: With diphenylphosphoranyl azide; 1,8-diazabicyclo[5.4.0]undec-7-ene in tetrahydrofuran T=20°C; 4 h; 2: With lithium aluminium tetrahydride in tetrahydrofuran T=20°C; 96 h;
参考文献
PROXIMAGEN LTD.; BOYD, Joe William; MEO, Paul; HIGGINBOTTOM, Michael; SIMPSON, Iain; MOUNTFORD, David Mark; SAVORY, Edward Daniel
Patent: WO2012/101453 A1, 2012 ;
Location in patent: Page/Page column 29-30 ;
WO 2012/101453 A1
