1: With sodium tetrahydroborate in methanol 3 h; 2: With hydrogenchloride; water in methanol; ethyl acetate 3: With sodium hydrogencarbonate in water; ethyl acetate
参考文献
PFIZER INC.
Patent: WO2006/106423 A2, 2006 ;
Location in patent: Page/Page column 33 ;
WO 2006/106423 A2