反应条件
1: 3-amino-pyrazole-4-carbonitrile With potassium carbonate in N,N-dimethyl-formamide T=0°C; 0.75 h; 2: methyl halide in N,N-dimethyl-formamide T=90°C; 10 h;
参考文献
Venkatesan, Gopalakrishnan; Paira, Priyankar; Cheong, Siew Lee; Vamsikrishna, Kosaraju; Federico, Stephanie; Klotz, Karl-Norbert; Spalluto, Giampiero; Pastorin, Giorgia
Bioorganic and Medicinal Chemistry, 2014 , vol. 22, # 5 p. 1751 - 1765