反应条件
1: sulfuric acid / 24 h / 80 °C 2: potassium carbonate / N,N-dimethyl-formamide / 0 - 20 °C 3: dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct; potassium acetate / N,N-dimethyl-formamide / 1.5 h / 100 °C / Microwave irradiation View Scheme
参考文献
Innocenti, Paolo; Cheung, Kwai-Ming J.; Solanki, Savade; Mas-Droux, Corine; Rowan, Fiona; Yeoh, Sharon; Boxall, Kathy; Westlake, Maura; Pickard, Lisa; Hardy, Tara; Baxter, Joanne E.; Aherne, G. Wynne; Bayliss, Richard; Fry, Andrew M.; Hoelder, Swen
Journal of Medicinal Chemistry, 2012 , vol. 55, # 7 p. 3228 - 3241