反应条件
1: HCl, isoamyl nitrite / dimethylformamide; dioxane / 0.17 h / -30 °C 2: Et3N / dimethylformamide / -20 °C / pH 8 3: 68 percent / TFA, 1,2-ethanedithiol / dimethylformamide / 0.25 h / 0 °C View Scheme
参考文献
Ishikawa, Kiyofumi; Fukami, Takehiro; Nagase, Toshio; Fujita, Kagari; Hayama, Takashi; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 11 p. 2139 - 2142