反应条件
ammonium chloride; O-(1H-benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium hexafluorophosphate; triethylamine in N,N-dimethyl-formamide T=0 - 20°C;
参考文献
LG LIFE SCIENCES LTD.; CHOI, Sung Pil; KIM, Geun Tae; SONG, Jeong Uk; KIM, Tae Hun; LIM, Dong Chul; KANG, Seung Wan; KIM, Hyung Jin
Patent: WO2010/93191 A2, 2010 ;
Location in patent: Paragraph 376-380 ;
WO 2010/093191 A2