反应条件
1: mercapto acetic acid ethylester With sodium hydride in tetrahydrofuran T=25°C; 2: (E)-2-Phenyl-3-chloro-4,4,4-trifluoro-but-2-en-1-al in tetrahydrofuran T=20°C; 20 h;
参考文献
Hale, Jeffrey J.; Lynch, Christopher L.; Neway, William; Mills, Sander G.; Hajdu, Richard; Keohane, Carol Ann; Rosenbach, Mark J.; Milligan, James A.; Shei, Gan-Ju; Parent, Stephen A.; Chrebet, Gary; Bergstrom, James; Card, Deborah; Ferrer, Marc; Hodder, Peter; Strulovici, Berta; Rosen, Hugh; Mandala, Suzanne
Journal of Medicinal Chemistry, 2004 , vol. 47, # 27 p. 6662 - 6665