反应条件
1: POCl3, N,N-dimethylaniline / toluene / 3 h / Heating 2: toluene / 3 h / Heating 3: 73 percent / EtSH, AlCl3 / 4 h / Ambient temperature View Scheme
参考文献
Liao, Yi; DeBoer, Peter; Meier, Eddie; Wikstroem, Hakan
Journal of Medicinal Chemistry, 1997 , vol. 40, # 25 p. 4146 - 4153