1: tetrahydrofuran / 2 h
2: H2O / 10 h / 40 °C
3: pyridine / CH2Cl2 / Ambient temperature
View Scheme
参考文献
Barbachyn, Michael R.; Hutchinson, Douglas K.; Brickner, Steven J.; Cynamon, Michael H.; Kilburn, James O.; et al.
J. Med. Chem., 1996 , vol. 39, # 3 p. 680 - 685