1: With dimethylsulfide borane complex in tetrahydrofuran T=0°C; 5 h; Heating / reflux; 2: With hydrogenchloride; water in tetrahydrofuran T=20°C; 3: With sodium hydrogencarbonate in water
参考文献
ASTRAZENECA AB
Patent: WO2006/73366 A1, 2006 ;
Location in patent: Page/Page column 200 ;
WO 2006/073366 A1