1: Harmine With sodium hydride in tetrahydrofuran; N,N-dimethyl-formamide T=20°C; 2: benzyl bromide in tetrahydrofuran; N,N-dimethyl-formamide 8 h; Heating / reflux; 3: With hydrogenchloride; sodium hydrogencarbonate more than 3 stages;
参考文献
Xinjiang Huashidan Pharmaceutical Research Co., Ltd.
Patent: EP1634881 A1, 2006 ;
Location in patent: Page/Page column 10; 11; 95 ;