1: With (benzotriazo-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in tetrahydrofuran 0.0833333 h; 2: With sodium tetrahydroborate in tetrahydrofuran T=20°C; 0.333333 h; 3: With hydrogenchloride; water in tetrahydrofuran; diethyl ether
参考文献
MERCK and CO., INC.
Patent: WO2006/102067 A1, 2006 ;
Location in patent: Page/Page column 34-35 ;