反应条件
1: With n-butyllithium; N,N,N',N,-tetramethylethylenediamine in diethyl ether T=-78 - 10°C; 2 h; 2: With N-fluoro-N-(phenylsulfonyl)benzene-sulfonamide in tetrahydrofuran; diethyl ether T=-70 - 0°C; 1 h;
参考文献
Hughes, Robert O.; Rogier, D. Joseph; Jacobsen, E. Jon; Walker, John K.; Maclnnes, Alan; Bond, Brian R.; Zhang, Lena L.; Yu, Ying; Zheng, Yi; Rumsey, Jeanne M.; Walgren, Jennie L.; Curtiss, Sandra W.; Fobian, Yvette M.; Heasley, Steven E.; Cubbage, Jerry W.; Moon, Joseph B.; Brown, David L.; Acker, Brad A.; Maddux, Todd M.; Tollefson, Mike B.; Mischke, Brent V.; Owen, Dafydd R.; Freskos, John N.; Molyneaux, John M.; Benson, Alan G.; Blevis-Ba, Rhadika M.
Journal of Medicinal Chemistry, 2010 , vol. 53, # 6 p. 2656 - 2660