反应条件
1: 98 percent / 1 N HCl / CHCl3 2: 1.) CDI, 2.) Et3N / 1.) THF, RT, 2 h, 2.) THF, RT 3: KOH, HONH2*HCl / methanol / Ambient temperature View Scheme
参考文献
Levy, Daniel E.; Lapierre, France; Liang, Weisheng; Ye, Wenqing; Lange, Christopher W.; Li, Xiaoyuan; Grobelny, Damian; Casabonne, Marie; Tyrrell, David; Holme, Kevin; Nadzan, Alex; Galardy, Richard E.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 2 p. 199 - 223
