反应条件
1: NaOH, H2O / dioxane; methanol / 0.5 h / Ambient temperature 2: HCl, H2O, TEA / acetonitrile / 0.5 h View Scheme
参考文献
Jahnsen, Rasmus D.; Frimodt-Moller, Niels; Franzyk, Henrik
Journal of Medicinal Chemistry, 2012 , vol. 55, # 16 p. 7253 - 7261