反应条件
1: 95 percent / hydrogen / Pd/C / ethyl acetate / 5 h / 20 °C 2: 79 percent / Na2CO3 / H2O; methanol / 12 h / 20 °C 3: 87 percent / EDAC; HOBt; DIPEA / dimethylformamide; CH2Cl2 / 12 h / 20 °C 4: 95 percent / hydrogen / Pd/C / methanol / 3 h / 20 °C 5: 85 percent / TFA / CH2Cl2 / 12 h / 20 °C View Scheme
参考文献
Righi, Giuliana; D'Achille, Claudia; Pescatore, Giovanna; Bonini, Carlo
Tetrahedron Letters, 2003 , vol. 44, # 37 p. 6999 - 7002