7-氯-1,3-二氢-5-(4-羟基苯基)-2H-1,4-苯并二氮杂卓-2-酮合成路线 (共 2 条)
反应条件
ammonia in ethanol; acetone
参考文献
Hoffmann-La Roche Inc.
Patent: US4191738 A1, 1980 ;
反应条件
mouse liver microsomes; NADPH; magnesium chloride in water aromatic hydroxylation; pH=7.4; 0.0666667 h; Enzyme kinetics;
参考文献
St-Pierre; Pang
Journal of Pharmacokinetics and Biopharmaceutics, 1995 , vol. 23, # 3 p. 243 - 266