反应条件
1.1: 78 percent / NaH / dimethylformamide / 20 °C
2.1: CH2Cl2 / 2 h / 20 °C
2.2: 75 percent / 1,1,1,3,3,3-hexamethyldisilazane / CH2Cl2 / 20 °C
View Scheme
参考文献
Smart, Brian P.; Oslund, Rob C.; Walsh, Laura A.; Gelb, Michael H.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 10 p. 2858 - 2860