(R)-(1-(4-((1H-吡咯并[2,3-B]吡啶-4-基)氨基甲酰)苯基)乙基)氨基甲酸苄酯合成路线 (共 1 条)
反应条件
1: With N-ethyl-N,N-diisopropylamine in acetonitrile T=20°C; 1 h; 2: With sodium methylate in methanol T=20°C; 0.5 h;
参考文献
Mitsubishi Pharma Corporation
Patent: EP1195372 A1, 2002 ;
Location in patent: Page 52-53 ;