反应条件
1: KOH / ethanol / 80 °C 2: 1-hydroxybenzotriazole, dicyclohexylcarbodiimide, N-methylmorpholine, Et3N / tetrahydrofuran; acetonitrile View Scheme
参考文献
Giardina, Giuseppe A. M.; Raveglia, Luca F.; Grugni, Mario; Sarau, Henry M.; Farina, Carlo; Medhurst, Andrew D.; Graziani, Davide; Schmidt, Dulcie B.; Rigolio, Roberto; Luttmann, Mark; Cavagnera, Stefano; Foley, James J.; Vecchietti, Vittorio; Hay, Douglas W. P.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 6 p. 1053 - 1065