2-甲氧基-6-(三氟甲基)嘧啶-4-醇合成路线 (共 2 条)
反应条件
sulfuric acid T=70°C; 2 h;
参考文献
Felczak, Krzysztof; Drabikowska, Alicja K.; Vilpo, Juhani A.; Kulikowski, Tadeusz; Shugar, David
Journal of Medicinal Chemistry, 1996 , vol. 39, # 8 p. 1720 - 1728
反应条件
thionyl chloride; N,N-dimethyl-formamide in toluene
T=80°C; 4 h;
参考文献
SUMITOMO CHEMICAL COMPANY, LIMITED; MIZUNO, Hajime
Patent: WO2010/134478 A1, 2010 ;
Location in patent: Page/Page column 178 ;